C1108Level 5
Gabapentin
**Semantic type:** Organic Chemical|Pharmacologic Substance
**Definition:** A synthetic analogue of the neurotransmitter gamma-aminobutyric acid with anticonvulsant activity. Although its exact mechanism of action is unknown, gabapentin appears to inhibit excitatory neuron activity. This agent also exhibits analgesic properties. (NCI04)
**Synonyms:** - 1-(aminomethyl)cyclohexaneacetic Acid - GABAPENTIN - Gralise - Neurontin - gabapentin
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