Saxagliptin

**Semantic type:** Pharmacologic Substance

**Definition:** A potent, selective and competitive, cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Saxagliptin is metabolized into an, although less potent, active mono-hydroxy metabolite.

**Synonyms:** - BMS-477118-11 - SAXAGLIPTIN - Saxagliptin Hydrate - Saxagliptin Monohydrate