C78130Level 6
Tolbutamide Sodium
**Semantic type:** Pharmacologic Substance
**Definition:** The sodium salt form of tolbutamide, a short-acting, first-generation sulfonylurea with hypoglycemic activity. Compared to second-generation sulfonylureas, tolbutamide is more likely to cause adverse effects, such as jaundice. This agent is rapidly metabolized by CYPC29.
**Synonyms:** - Orinase - TOLBUTAMIDE SODIUM
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