C81529Level 5
Dalcetrapib
**Semantic type:** Pharmacologic Substance
**Definition:** A cholesteryl ester transfer protein (CETP) inhibitor that can produce an increase in serum HDL-cholesterol levels and a decrease in serum LDL-cholesterol levels. Dalcetrapib is structurally dissimilar from other CETP inhibitors, including torcetrapib, and raises functional HDL by a different mechanism.
**Synonyms:** - DALCETRAPIB - R1658
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