C81702Level 6
Saxagliptin Hydrochloride
**Semantic type:** Pharmacologic Substance
**Definition:** The hydrochloride salt form of saxagliptin, an orally bioavailable, potent, selective and competitive, cyanopyrrolidine-based inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Saxagliptin is metabolized into an, although less potent, active mono-hydroxy metabolite.
**Synonyms:** - SAXAGLIPTIN HYDROCHLORIDE
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